Discovery of small-molecule inhibitors of Uba1 and development of step-specific assays for PCNA ubiquitination

Gaur Paras
2020

Unraveling the Mechanism of Action of Myricetin in the Inhibition of hUba1∼Ubiquitin Thioester Bond Formation via In Silico Molecular Modeling Techniques

Gaur Paras, Tyagi Chetna
2023

Mode of inhibitory binding of epigallocatechin gallate to the ubiquitin-activating enzyme Uba1 via accelerated molecular dynamics

Gaur Paras, Fenteany Gabriel, Tyagi Chetna
2021

Robust high-throughput assays to assess discrete steps in ubiquitination and related cascades

Fenteany Gabriel, Gaur Paras, Sharma Gaurav, Pintér Lajos, Kiss Ernő, Haracska Lajos
2020

A series of xanthenes inhibiting Rad6 function and Rad6–Rad18 interaction in the PCNA ubiquitination cascade

Fenteany Gabriel, Sharma Gaurav, Gaur Paras, Borics Attila, Wéber Edit, Kiss Ernő, Haracska Lajos
2022

Multilevel structure–activity profiling reveals multiple green tea compound families that each modulate ubiquitin-activating enzyme and ubiquitination by a distinct mechanism

Fenteany Gabriel, Gaur Paras, Hegedűs Lili, Dudás Kata, Kiss Ernő, Wéber Edit, Hackler László, ifj, Martinek Tamás A., Puskás László, Haracska Lajos
2019